Publications

General literature

DOI

Boehringer Ingelheim experiments with open-access chemical probes

A. Mullard Boehringer Ingelheim experiments with open-access chemical probes, Nature Reviews Drug Discovery 2018, 17, 7.

Molecule specific literature

Enzyme
DOI

HIV NNRTI | BI-2540

Practical Synthesis of A Benzophenone-Based NNRT Inhibitor of HIV-1

Xiao-jun Wang, Li Zhang, Xiufeng Sun, Heewon Lee, Dhileepkumar Krishnamurthy, Jeff A. O’Meara, Serge Landry, Christiane Yoakim, Bruno Simoneau, Nathan K. Yee, and Chris H. Senanayake

Org. Process Res. Dev. 2012, 16, 561-566.

Enzyme
DOI
PUBMED

HIV NNRTI | BI-2540

Peris Non-nucleoside reverse transcriptase inhibitors: a review on pharmacokinetics, pharmacodynamics, safety and tolerability

Iris Usach, Virginia Melis and Jose-Esteban Peris

J. Int AIDS Soc. 2013, 16, 1-14.

Enzyme
DOI
PUBMED

HIV NNRTI | BI-2540

Structure and function of HIV-1 reverse transcriptase: molecular mechanisms of polymerization and inhibition

Stefan G. Sarafianos, Bruno Marchand, Kalyan Das, Daniel M. Himmel, Michael A. Parniak, Stephen H. Hughes and Eddy Arnold

J. Mol Biol. 2009, 385, 693-713.